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Epigenetics
Epigenetics
♦HDAC
(
0
)
ITSA-1
Tubastatin A TFA
SR-4370
Tinostamustine
BML-210 (CAY10433)
Suprastat
NR-160
Quisinostat HCl
NKL 22
HDAC-IN-7
SS-208
Sodium Butyrate
♦HIF
(
0
)
Roxadustat (FG-4592)
IOX2
BAY 87-2243
PX-478 2HCl
FG-2216 (YM-311; IOX-3; YM-311)
KC7F2
MK-8617
♦ PARP
(
0
)
♦JAK
(
0
)
Itacitinib (INCB-039110)
Itacitinib adipate (INCB 39110 adipate)
Ruxolitinib Phosphate (INC-424, INCB-18424, INCB-018424, Jakafi and Jakavi)
Ruxolitinib sulfate (INC 424, INCB 18424, INCB 018424, Jakafi, Jakavi)
Baricitinib phosphate (LY-3009104, INCB-028050, Olumiant)
Ruxolitinib (INCB-018424; INC-424)
Tofacitinib (CP690550) Citrate
AZD1480
Fedratinib (SAR302503)
AT9283
BMS-911543
Decernotinib (VX-509; VRT-831509; adelatinib)
Peficitinib (ASP-015K, JNJ-54781532)
AG-490 (Tyrphostin B42; zinc0255794)
Momelotinib (LM1149; CYT387; CYT11387)
FLLL32
Cerdulatinib HCl (PRT-2070; PRT-062070)
Filgotinib (GLPG-0634)
Go6976 (PD40697)
GLPG0634 analogue
ZM 39923 HCl
XL019
Pacritinib (SB1518)
Curcumol
CEP-33779
AZ 960
NVP-BSK805 2HCl (BSK-805)
S-Ruxolitinib (INCB-018424)
Baricitinib (LY-3009104, INCB-028050)
Gandotinib (LY-2784544)
Tofacitinib (CP690550; tasocitinib)
G5-7
Oclacitinib maleate (PF-03394197)
Cerdulatinib
Solcitinib (GSK2586184; GLPG-0778)
Pyridone 6
SAR-20347
CHZ868
Oclacitinib (PF-03394197)
PF-06700841 tosylate
WHI-P97
JAK3-IN-6
Abrocitinib (PF04965842)
Upadacitinib tartrate
FM-479
(3S,4S)-Tofacitinib
JAK1-IN-4
Protosappanin A
TCJL-37
Fedratinib (TG101348) dihydrochloride hydrate
Delgocitinib (LEO124249; JTE052)
Ilginatinib (NS-018)
Golidocitinib (AZD-4205)
NVP-BSK805
(3S,4R)-Tofacitinib
(3R,4S)-Tofacitinib
♦Aurora Kinase
(
0
)
Alisertib (MLN8237, MLN-8237)
Tozasertib (VX680; MK0457)
Barasertib ( INH-34; AZD-1152-HQPA)
ZM 447439
MLN8054
Danusertib (PHA739358)
BI-847325
MK-8745
KW-2449
JNJ-7706621
GSK1070916 (NMI900 or GSK1070916 A)
CCT137690
MK-5108 (VX689)
TCS7010 (Aurora A Inhibitor I)
CCT129202
PHA-680632
Hesperadin
TAK-901
ENMD-2076
CYC116
AMG-900
PF-03814735
SNS-314 Mesylate
SNS-314
♦Histone Acetyltransferase
(
0
)
Ranolazine (CVT303, RS43285-003; Ranexa)
Remodelin
WM 3835
C646
MG149
Remodelin HBr
Anacardic Acid (Hydroginkgolic acid)
I-CBP112
CTB
WM-1119
TTK21
A-485
Curcumin
WM-8014
♦Histone Demethylase
(
0
)
OG-L002
JIB-04 (NSC-693627)
IOX1
SP2509 (HCI-2509)
Iadademstat (ORY-1001; RG6016) 2HCl
ML324 (CID44143209)
GSK-LSD1 2HCl
CPI-455
GSK-J4
DDP-38003 dihydrochloride
AS8351
NCGC00244536
GSK-690
GSK2879552
Seclidemstat
GSK2807 TFA
GSK J4 HCl
T-3775440 HCl
Pulrodemstat (CC90011)
CBB1007
Furazolidone
KDM5-IN-48
JIB-04 Z-isomer
KDM5-C70
PBIT
Procaine (Novocaine)
Pulrodemstat (CC90011) besylate
GSK-690 HCl
♦Histone Methyltransferase
(
0
)
Pinometostat (EPZ-5676)
EPZ005687
GSK343
BIX 01294
Tazemetostat (EPZ6438; E-7438)
SGC707
3-deazaneplanocin A (DZNeP; NSC 617989) HCl
UNC1999
CPI-360
GSK503
AMI-1 disodium salt
CPI-169
EPZ015666 (GSK3235025)
GSK126 (GSK2816126; GSK 2816126A)
UNC0379
EI1 (KB145943; EI 1)
BRD4770
UNC0631
PFI-2
MI-3
SGC 0946
MM-102
EPZ004777
Entacapone (OR611)
UNC1215
5WKS
UNC0646
SGC2085 HCl
ZINC30303842
Dot1L-IN-4
PFI-2 HCl
EPZ020411
UNC0638
MS049 2HCl
UNC3866
Lirametostat (CPI-1205)
OICR-9429
SGC2085
HLCL-61(HCl)
C-7280948
EPZ015866 (GSK591; GSK3203591)
MS023
A-196
CM-272
JQ-EZ-05 (JQEZ5)
UNC0642
LLY-283
GSK3326595 (EPZ-015938)
BIX01294 triHCl
UNC0224
UNC0321
BIX01338
BRD9539
Chaetocin
Sinefungin
EBI-2511
BAY-598
Onametostat (JNJ-64619178)
BCI-121
Amodiaquin HCl hydrate
A-366
AZ-505 2TFA salt
TP-064
DCLX069
DS-437
EPZ011989
EPZ031686
EZM2302 (GSK-3359088)
Urea J Acid
MM-401
LLY-507
MAK-683
MI-503
Valemetostat
WDR5-0103
XY1
EPZ020411 hydrochloride
MS023 dihydrochloride
MM-102 TFA
Valemetostat tosylate
GSK3368715
GSK3368715 dihydrochloride
EPZ004777 hydrochloride
MS049
CMP-5
MS1943
UNC6852
♦ DNA Methyltransferase
(
0
)
Levetiracetam (UCB-L 059, SIB-S 1)
Decitabine (NSC-127716)
Azacitidine (Ladakamycin; 5-AzaC)
RG108
Thioguanine (NSC-752; Tabloid)
Zebularine (NSC309132; 4-Deoxyuridine)
SGI-1027
Lomeguatrib (PaTrin2)
Procainamide HCl
(-)-Epigallocatechin Gallate
BOBCAT339
Bobcat339 HCl
DC_05
GSK-3484862
♦Epigenetic Reader Domain
(
0
)
UNC-926
MI-2 (Menin-MLL Inhibitor)
(+)-JQ1
I-BET151 (GSK1210151A)
PFI-1 (PF-6405761)
Molibresib (I-BET762; GSK-525762A)
Apabetalone (RVX-08, RVX-000222)
PFI-4
SGC-CBP30
Bromosporine
GSK2801 (GSK-2801)
OF-1 (OF-1)
MS436
GSK1324726A (I-BET-726)
PFI-3
CPI-203 (RO-6870810, TEN-010, JQ2, and RG-6146)
Birabresib (OTX015; MK8628)
UNC669
PF-CBP1 HCl
GSK620
PF-CBP1
BRM/BRG1 ATP Inhibitor-1
Menin-MLL inhibitor 20
MI-463
CPI-637
CPI-0610
EED226
GSK9311
GSK6853
AZD5153 HNT salt
BI-9564
Mivebresib
PLX51107
PF-CBP1
BMS-986158
GSK4028
ARV-825
BETd-246
KG-501
(+)-JQ1 carboxylic acid
(+)-JQ1 PA
INCB057643
INCB054329
ZL0420
ZL0454
GSK-5959
BAY-299
BAY-850
BAY-1238097
(R)-BAY1238097
BET-BAY 002 S enantiomer
GNE-272
GNE-781
ABBV-744
BI-7273
666-15
BI-894999
CPI-268456
dBET57
IACS-9571
I-BRD9
NI-57
Y06036
Y06137
Inobrodib (CCS1477)
FL-411
Molibresib besylate
MI-136
Bromodomain inhibitor-8
I-BET762 carboxylic acid
Thalidomide-NH-C4-NH-Boc
TP-472
♦Sirtuin
(
0
)
SRT1720 HCL (CAY-10559)
Selisistat (SEN0014196; EX 527)
Resveratrol (SRT501; RM1812)
Sirtinol
Nicotinamide (Vitamin B3)
Fisetin (Fustel; CCRIS-9034; NSC-407010)
AGK2
Splitomicin (Splitomycin)
SRT2104 (GSK-2245840)
SirReal2
CAY10602
SRT3025 HCL
OSS-128167
Cambinol
SRT1720
AK-7
AK-1
Lithospermic acid B
SIRT7 inhibitor 97491
♦Pim
(
0
)
SGI-1776
(Z)-SMI-4a
AZD1208
CX-6258 HCl
CX-6258
PIM447
♦PKC
(
0
)
PKC-theta inhibitor
Ruboxistaurin hydrochloride (LY333531)
LXS196
CHELERYTHRINE CHLORIDE
CMPD-101
R59022
Ruboxistaurin (LY333531)
Ingenol
Protein kinase inhibitor H-7
Verbascoside (Acteoside; Kusaginin; TJC160)
TPPB
Phorbol 12,13-dibutyrate
PKCß inhibitor
Chelerythrine
VTX-27
D-erythro-Sphingosine (Erythrosphingosine)
N-Desmethyltamoxifen HCl
♦SMYD
(
0
)
AZ505 free base
♦MAT
(
0
)
FIDAS-5
AG-270
PF-9366
MAT2A inhibitor 2
FIDAS-5
♦MicroRNA
(
0
)
Targapremir-210 (TGP-210)
LIN28 inhibitor LI71
♦AMPK
(
0
)
ASP4132 tosylate
BC1618
Marein
Buformin hydrochloride
Ginkgolide C (BN-52022)
IM156 acetate (HL156A; Lixumistat; HL271)
♦Protein Arginine Deiminase
(
0
)
GSK484
Cl-amidine
BB-Cl-Amidine
♦EZH1/2
(
0
)
PF-06726304
♦MLL
(
0
)
SNDX-5613
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