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Protein Tyrosine Kinase
Protein Tyrosine Kinase
♦VEGFR
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Sunitinib Malate (SU-11248 Malate)
Cabozantinib (XL184; BMS907351; Cometriq)
Ponatinib (AP-24534; Iclusig)
Axitinib (AG-013736; Inlyta)
Foretinib (GSK-1363089; XL-880; EXEL2880; GSK-089)
Vandetanib (ZD-6474)
SU5402 (SU-5402; SU 5402)
AZD2932
Sunitinib free base (SU-11248)
Dovitinib (TKI258; CHIR-258 ) Lactate
LY2874455
SKLB1002 (SKLB-1002; SKLB 1002)
BMS-794833
Ki8751
Apatinib (Rivoceranib, YN968D1)
Tivozanib (AV951; KRN-951)
Brivanib (BMS-540215)
Dovitinib (TKI-258, CHIR-258)
Lenvatinib (E7080; ER-203492-00)
OSI-930
Pazopanib HCl (GW-786034; GW786034; Votrient)
RAF265 (CHIR-265)
Brivanib Alaninate (BMS-582664)
PD173074
Pazopanib (GW 786034; Votrient)
Vatalanib (PTK-787; ZK222584; CGP79787) 2HCl
Dovitinib Dilactic Acid (TKI258; CHIR258)
Cediranib (NSC-732208; AZD-2171)
Orantinib (SU 6668; NSC-702827; TSU68)
MGCD-265 analog
SAR131675
Semaxanib (SU-5416)
ZM 323881 HCl
Golvatinib (E7050)
ZM 306416 (CB676475)
Cabozantinib malate (XL184)
KRN 633
ENMD-2076 Tartrate
Linifanib (ABT-869; AL-39324)
Nintedanib (Vargatef; BIBF 1120)
Motesanib Diphosphate (AMG-706)
Telatinib (BAY 57-9352)
BFH772
Cediranib maleate
Apatinib mesylate
Telatinib mesylate (Bay 57-9352 mesylate)
♦EGFR
(
0
)
Chrysophanic Acid (Chrysophanol)
WHI-P154
AEE788 (NVP-AEE788)
Erlotinib HCl (OSI-744, Tarceva)
Gefitinib (ZD 1839)
Lapatinib Ditosylate (GW-572016, Tykerb)
Afatinib (BIBW2992)
Neratinib (HKI-272; PB272; Nerlynx)
Neratinib (HKI-272; PB272; Nerlynx)
Zorifertinib (AZD3759; AZD-3759; zorifertinibum)
Canertinib (CI-1033; PD-183805)
Lapatinib (GW-572016, Tykerb, Tyverb)
AZ5104
Afatinib (BIBW2992) Dimaleate
CL-387785 (EKI-785)
Erlotinib (OSI744, Tarceva)
Poziotinib (HM781-36B)
Osimertinib (AZD9291; Tagrisso)
PD168393 (PD-168393)
CNX-2006
AG-18 (RG50858, TX-825)
Butein (NSC-652892; CCG208298; CS-5675; AC 1NQY7L)
Rociletinib (CO-1686, AVL-301, CNX-419)
WZ4002
Pelitinib (EKB-569; WAY-EKB 569)
AC480 (BMS599626)
TAK-285
CP-724714
Dacomitinib (PF-299804, PF-299)
AG-1478 (Tyrphostin AG-1478; NSC693255)
Allitinib (AST 1306)
OSI-420 (Desmethyl Erlotinib) HCl
Tyrphostin 9 (AG17; Malonoben)
WZ3146
WZ8040
Sapitinib (AZD-8931)
PD153035 HCl (SU5271; ZM252868)
Icotinib (BPI2009)
Varlitinib (ARRY-543; ARRY-334543; ASLAN-001)
Genistein (NPI031L; BIO-00; G2535; PTI G-4660; SIPI9764I)
Nazartinib (EGF816, NVS-816)
♦ PDGFR
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0
)
Imatinib (STI571; Gleevec; Glivec)
Tyrphostin AG 1296
MK-2461
Masitinib (AB1010)
CP-673451
Sennoside B
Amuvatinib (MP470; HPK56)
Crenolanib (CP-868596; RO 002; ARO 002)
Ripretinib (DCC-2618)
Anlotinib
Anlotinib Dihydrochloride
♦c-MET
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0
)
Crizotinib (Xalkori; PF02341066)
PHA-665752
SU11274 (PKI SU11274; PKI SU11274)
SGX-523
BMS-777607 (BMS-817378; ASLAN-002)
Tepotinib (EMD 1214063)
NVP-BVU972
Capmatinib (INCB28060; INC-280)
AMG-208
AMG-458
JNJ-38877605
BMS-754807
PF-04217903
Tivantinib (ARQ 197)
♦ HER-2
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0
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Mubritinib (TAK 165)
Tyrphostin AG 879
♦ALK
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0
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Alectinib HCl (ALECENSA, AF-802, CH-5424802, RO-5424802)
Ceritinib (LDK-378; Zykadia)
TAE684 (NVP-TAE684)
Alectinib (AF-802, CH-5424802, RO-5424802, Alecensa)
Brigatinib (AP26113)
GSK1838705A
Entrectinib (NMS-E 628; RXDX101; ROZLYTREK)
AZD3463
ASP3026
Loratinib (PF-06463922; Lorlatinib; lorbrena)
♦ FLT3
(
0
)
Tamatinib besylate (R406)
Quizartinib (AC220; AC010220)
Tandutinib (MLN518, CT53518, NSC-726292)
UNC-2025 HCl
AMG 925 (FLX925; AMG925)
G-749
TCS 359
UNC-2025
♦FGFR
(
0
)
Infigratinib (BGJ-398; NVP-BG-J398)
FIIN-2
AZD4547
BLU9931
CH5183284 (FF-284; Debio-1347)
SSR128129E (SSR 128129E; SSR128129 E)
BLU-554(BLU-554)
PD166866
ACTB-1003
Roblitinib (FGF 401)
♦IFG-1R
(
0
)
OSI-906 (Linsitinib)
NVP-AEW541
GSK1904529A (GSK-4529; GSK-1904529A; GSK 4529)
NVP-ADW742
BMS-536924 (CS0117; BMS 536924)
AG-1024 (Tyrphostin; Tyrphostin AG1024)
PQ 401
Picropodophyllin (Picropodophyllotoxin, AXL-1717 or PPP)
♦c-Kit
(
0
)
Imatinib Mesylate (STI571; Gleevec; Glivec)
Pexidartinib (PLX3397; Turalio; CML261; FP113)
Dasatinib Monohydrate (BMS354825; Sprycel)
♦ Tie-2
(
0
)
Tie2 kinase inhibitor
♦CSF-1R
(
0
)
GW2580 (SC203877)
BLZ945
♦TAM Receptor
(
0
)
NPS-1034
R428 (BGB-324; R-428)
UNC2250
UNC2881
LDC1267
Dubermatinib (TP-0903)
♦Trk receptor
(
0
)
GW441756
GNF-5837
ANA-12
♦c-RET
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0
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